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Structure: Internal structure identifier : 184933
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Identification of a novel quinoline-based DNA demethylating compound highly potent in cancer cells

Clemens Zwergel , Michael Schnekenburger , Federica Sarno , Cecilia Battistelli , Maria Cristina Manara , et al.
Clinical Epigenetics, 2019, 11 (1), pp.68. ⟨10.1186/s13148-019-0663-8⟩
Journal articles hal-02383678v1
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Novel Quinoline Compounds Active in Cancer Cells through Coupled DNA Methyltransferase Inhibition and Degradation

Clemens Zwergel , Rossella Fioravanti , Giulia Stazi , Federica Sarno , Cecilia Battistelli , et al.
Cancers, 2020, 12 (2), pp.447. ⟨10.3390/cancers12020447⟩
Journal articles pasteur-03026533v1
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Targeting DNA Methylation with Small Molecules: What’s Next?

Alexandre Erdmann , Ludovic Halby , Jacques Fahy , Paola B Arimondo
Journal of Medicinal Chemistry, 2015, 58 (6), pp.2569-2583. ⟨10.1021/jm500843d⟩
Journal articles hal-03043209v1
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Synthesis of novel 3-halo-3-nitroflavanones and their activities as DNA methyltransferase inhibitors in cancer cells

Dany Pechalrieu , Daniel Dauzonne , Paola Arimondo , Marie Lopez
European Journal of Medicinal Chemistry, 2020, pp.111829. ⟨10.1016/j.ejmech.2019.111829⟩
Journal articles hal-02394113v1
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Hemisynthetic alkaloids derived from trilobine are antimalarials with sustained activity in multidrug-resistant Plasmodium falciparum

Flore Nardella , Irina Dobrescu , Haitham Hassan , Fabien Rodrigues , Sabine Thiberge , et al.
iScience, 2023, 26 (2), pp.105940. ⟨10.1016/j.isci.2023.105940⟩
Journal articles pasteur-04099097v1
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New insights into the role of DNA methylation in Biomphalaria glabrata infection susceptibility

Nelia Luviano , Marie Lopez , Fleur Gawehns , Cristian Chaparro , Paola B Arimondo , et al.
XVI Symposium on Schistosomiasis, FIOCRUZ, Nov 2022, Ouro Preto, Brazil
Conference papers hal-03963335v1
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Demethylation by low-dose 5-aza-2′-deoxycytidine impairs 3D melanoma invasion partially through miR-199a-3p expression revealing the role of this miR in melanoma

Cécile Desjobert , Arnaud Carrier , Audrey Delmas , Diego Marzese , Antoine Daunay , et al.
Clinical Epigenetics, 2019, 11 (1), pp.9. ⟨10.1186/s13148-018-0600-2⟩
Journal articles hal-02332300v1
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Properly Substituted Analogues of BIX-01294 Lose Inhibition of G9a Histone Methyltransferase and Gain Selective Anti-DNA Methyltransferase 3A Activity

Dante Rotili , Domenico Tarantino , Biagina Marrocco , Christina Gros , Véronique Masson , et al.
PLoS ONE, 2014, 9 (5), pp.e96941. ⟨10.1371/journal.pone.0096941⟩
Journal articles pasteur-03182293v1
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Epigenetically regulated PCDHB15 impairs aggressiveness of metastatic melanoma cells

Arnaud Carrier , Cécile Desjobert , Valérie Lobjois , Lise Rigal , Florence Busato , et al.
Clinical Epigenetics, 2022, 14 (1), pp.156. ⟨10.1186/s13148-022-01364-x⟩
Journal articles pasteur-03946850v2
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DNA methylome combined with chromosome cluster-oriented analysis provides an early signature for cutaneous melanoma aggressiveness

Arnaud Carrier , Cécile Desjobert , Loic Ponger , Laurence Lamant , Matias Bustos , et al.
eLife, 2022, 11, pp.e78587. ⟨10.7554/eLife.78587⟩
Journal articles hal-03798060v1
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Bisubstrate-Type Chemical Probes Identify GRP94 as a Potential Target of Cytosine-Containing Adenosine Analogs

Dany Pechalrieu , Fanny Assemat , Ludovic Halby , Marlene Marcellin , Pengrong Yan , et al.
ACS Chemical Biology, 2020, 15 (4), pp.952-961. ⟨10.1021/acschembio.9b00965⟩
Journal articles pasteur-03026521v1