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From Substrate to Fragments to Inhibitor Active In Vivo against Staphylococcus aureus
Muriel Gelin
,
Julie Paoletti
,
Marie-Anne Nahori
,
Valeŕie Huteau
,
Clarisse Leseigneur
,
et al.
Journal articles
hal-02573173v1
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Diacylglyceride kinases, sphingosine kinases and NAD kinases: distant relatives of 6-phosphofructokinases
Gilles Labesse
,
Dominique Douguet
,
Liliane Assairi
,
Anne-Marie Gilles
Journal articles
istex
hal-02115578v1
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Comparative modelling and immunochemical reactivity of Escherichia coli UMP kinase
Gilles Labesse
,
Nadia Bucurenci
,
Dominique Douguet
,
Hiroshi Sakamoto
,
Stéphanie Landais
,
et al.
Journal articles
istex
hal-02115583v1
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Structure of the oncoprotein Rcl bound to three nucleotide analogues.
André Padilla
,
Claire Amiable
,
Sylvie Pochet
,
Pierre-Alexandre Kaminski
,
Gilles Labesse
Journal articles
pasteur-00796442v1
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Structural basis for the allosteric inhibition of UMP kinase from Gram‐positive bacteria, a promising antibacterial target
Patrick Walter
,
Ariel E Mechaly
,
Julien Bous
,
Ahmed Haouz
,
Patrick England
,
et al.
Journal articles
pasteur-04096367v1
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New Chemical Probe Targeting Bacterial NAD Kinase
David A. Clément
,
Clarisse Leseigneur
,
Muriel Gelin
,
Dylan Coelho
,
Valérie Huteau
,
et al.
Journal articles
hal-03030945v1
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First-in-class allosteric inhibitors of bacterial IMPDHs
Thomas Alexandre
,
Alexandru Lupan
,
Olivier Helynck
,
Sophie Vichier-Guerre
,
Laurence Dugué
,
et al.
Journal articles
pasteur-02125232v1
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