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authFullName_s : Ludovic Halby
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Towards the sustainable discovery and development of new antibiotics

Marcus Miethke , Marco Pieroni , Tilmann Weber , Mark Brönstrup , Peter Hammann , et al.
Nature Reviews Chemistry, 2021, 5 (10), pp.726-749. ⟨10.1038/s41570-021-00313-1⟩
Journal articles pasteur-03427787v1
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A novel screening strategy to identify histone methyltransferase inhibitors reveals a crosstalk between DOT1L and CARM1

Yang Si , Corentin Bon , Magdalena Barbachowska , Veronique Cadet-Daniel , Corinne Jallet , et al.
RSC Chemical Biology, 2022, 3 (4), pp.456-467. ⟨10.1039/d1cb00095k⟩
Journal articles pasteur-03693863v1
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Targeting DNA Methylation with Small Molecules: What’s Next?

Alexandre Erdmann , Ludovic Halby , Jacques Fahy , Paola B Arimondo
Journal of Medicinal Chemistry, 2015, 58 (6), pp.2569-2583. ⟨10.1021/jm500843d⟩
Journal articles hal-03043209v1
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An epigenetic molluscicide

Nelia Luviano , Ludovic Halby , Corinne Jallet , Paola B Arimondo , Celine Cosseau , et al.
Preprints, Working Papers, ... hal-04157076v1
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Editorial : Bisubstrate inhibitors: the promise of a selective and potent chemical inhibition of epigenetic “writers

Corentin Bon , Ludovic Halby , Paola B Arimondo , Paola B Arimondo
Epigenomics, 2020, 12 (17), pp.1479-1482. ⟨10.2217/epi-2020-0203⟩
Journal articles pasteur-03023370v1
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DNA Methylation Bisubstrate Inhibitors Are Fast-Acting Drugs Active against Artemisinin-Resistant Plasmodium falciparum Parasites

Flore Nardella , Ludovic Halby , Elie Hammam , Diane Erdmann , Véronique Cadet-Daniel , et al.
ACS Central Science, 2020, 6 (1), pp.16-21. ⟨10.1021/acscentsci.9b00874⟩
Journal articles hal-02571983v1

Espoirs et promesses de la méthylation de l’ADN et des histones comme cibles anticancéreuses

Corentin Bon , Diane Erdmann , Ludovic Halby , Paola B Arimondo
Bulletin du Cancer, 2019, 106 (10), pp.823-833. ⟨10.1016/j.bulcan.2019.08.001⟩
Journal articles hal-02383686v1
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Direct Synthesis of Allyl Amines with 2‐Nitrosulfonamide Derivatives via the Tsuji‐Trost Reaction

Corentin Bon , Paola B Arimondo , Ludovic Halby
ChemistryOpen, 2021, pp.Online Version of Record before inclusion in an issue. ⟨10.1002/open.202100147⟩
Journal articles pasteur-03411855v1
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Hemisynthetic alkaloids derived from trilobine are antimalarials with sustained activity in multidrug-resistant Plasmodium falciparum

Flore Nardella , Irina Dobrescu , Haitham Hassan , Fabien Rodrigues , Sabine Thiberge , et al.
iScience, 2023, 26 (2), pp.105940. ⟨10.1016/j.isci.2023.105940⟩
Journal articles pasteur-04099097v1
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New insights into the role of DNA methylation in Biomphalaria glabrata infection susceptibility

Nelia Luviano , Marie Lopez , Fleur Gawehns , Cristian Chaparro , Paola B Arimondo , et al.
XVI Symposium on Schistosomiasis, FIOCRUZ, Nov 2022, Ouro Preto, Brazil
Conference papers hal-03963335v1
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Procainamide-SAHA fused inhibitors of hHDAC6 tackle multi-drug resistant malaria parasites

Flore Nardella , Ludovic Halby , Irina Dobrescu , Johanna Viluma , Corentin Bon , et al.
Journal of Medicinal Chemistry, 2021, 64 (14), pp.10403-10417. ⟨10.1021/acs.jmedchem.1c00821⟩
Journal articles hal-03264653v1
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Quinazoline-based analog of adenine as an antidote against MLL-rearranged leukemia cells: synthesis, inhibition assays and docking studies

Corentin Bon , Magdalena Barbachowska , Nemanja Djokovic , Dusan Ruzic , Yang Si , et al.
Future Medicinal Chemistry, 2022, 14 (8), pp.557-570. ⟨10.4155/fmc-2021-0251⟩
Journal articles pasteur-03704094v1
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Bisubstrate-Type Chemical Probes Identify GRP94 as a Potential Target of Cytosine-Containing Adenosine Analogs

Dany Pechalrieu , Fanny Assemat , Ludovic Halby , Marlene Marcellin , Pengrong Yan , et al.
ACS Chemical Biology, 2020, 15 (4), pp.952-961. ⟨10.1021/acschembio.9b00965⟩
Journal articles pasteur-03026521v1
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Synthesis and Biological Activity of a Cytostatic Inhibitor of MLLr Leukemia Targeting the DOT1L Protein

Corentin Bon , Yang Si , Melanie Pernak , Magdalena Barbachowska , Eva Levi-Acobas , et al.
Molecules, 2021, Special Issue The Chemical Biology Research in France, 26 (17), pp.5300. ⟨10.3390/molecules26175300⟩
Journal articles pasteur-03411876v1