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Mycobacterium tuberculosis thymidine monophosphate kinase inhibitors: Biological evaluation and conformational analysis of 2 '- and 3 '-modified thymidine analogues
Philippe van Rompaey
,
Koen Nauwelaerts
,
Veerle Vanheusden
,
Jef Rozenski
,
Hélène Munier-Lehmann
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et al.
Journal articles
pasteur-00167037v1
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A short path synthesis of [13C/15N] multilabeled pyrimidine nucleosides starting from glucopyranose nucleosides.
Irene M Lagoja
,
Sylvie Pochet
,
Valerie Boudou
,
Roy Little
,
Eveline Lescrinier
,
et al.
Journal articles
istex
pasteur-00166200v1
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Noncanonical DNA polymerization by aminoadenine-based siphoviruses
Valerie Pezo
,
Faten Jaziri
,
Pierre-Yves Bourguignon
,
Dominique Louis
,
Deborah Jacobs-Sera
,
et al.
Journal articles
pasteur-03228903v1
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Structural Studies of HNA Substrate Specificity in Mutants of an Archaeal DNA Polymerase Obtained by Directed Evolution
Camille Samson
,
Pierre Legrand
,
Mustafa Tekpinar
,
Jef Rozenski
,
Mikhail Abramov
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et al.
Journal articles
pasteur-03269775v1
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Synthesis and evaluation of 6-aza-2'-deoxyuridine monophosphate analogs as inhibitors of thymidylate synthases, and as substrates or inhibitors of thymidine monophosphate kinase in Mycobacterium tuberculosis.
Martin Kögler
,
Roger Busson
,
Steven de Jonghe
,
Jef Rozenski
,
Kristien van Belle
,
et al.
Journal articles
pasteur-00705897v1
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Discovery of bicyclic thymidine analogues as selective and high-affinity inhibitors of Mycobacterium tuberculosis thymidine monophosphate kinase.
Veerle Vanheusden
,
Hélène Munier-Lehmann
,
Matheus Froeyen
,
Roger Busson
,
Jef Rozenski
,
et al.
Journal articles
pasteur-00166959v1
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